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Cytochrome P450 3A5 Inhibitors [MoA] Mechanism of Action Drugs

NDC Number Brand Name Generic Name Labeler Dosage Form DEA Schedule Marketing Start Date
0024-4512 Fexinidazole Fexinidazole Sanofi-Aventis U.S. LLC TABLET 2021-07-16
0093-3219 Ketoconazole Ketoconazole Teva Pharmaceuticals USA, Inc. CREAM 2019-02-08
0168-0099 ketoconazole ketoconazole E. Fougera & Co. a division of Fougera Pharmaceuticals Inc. CREAM 2004-04-28
0713-0592 Ketoconazole Ketoconazole Cosette Pharmaceuticals, Inc. SHAMPOO, SUSPENSION 2025-02-07
16714-955 Ketoconazole Ketoconazole NORTHSTAR RX LLC CREAM 2002-12-18
21922-025 Ketoconazole Ketoconazole Cream, 2% Encube Ethicals, Inc. CREAM 2021-05-27
35573-433 KETOCONAZOLE ketoconazole Burel Pharmaceuticals, LLC TABLET 2020-04-10
43538-530 Ketodan ketoconazole Medimetriks Pharmaceuticals, Inc. AEROSOL, FOAM 2012-06-15
45802-465 Ketoconazole Ketoconazole Padagis Israel Pharmaceuticals Ltd SHAMPOO, SUSPENSION 2010-01-19
45802-532 ketoconazole ketoconazole Padagis Israel Pharmaceuticals Ltd AEROSOL, FOAM 2011-08-30
50090-3288 Ketoconazole Ketoconazole A-S Medication Solutions SHAMPOO, SUSPENSION 2005-04-11
50090-5265 Ketoconazole Ketoconazole A-S Medication Solutions CREAM 2019-02-08
50090-6046 Ketoconazole Ketoconazole Cream, 2% A-S Medication Solutions CREAM 2021-05-27
50090-6069 Ketoconazole Ketoconazole A-S Medication Solutions CREAM 2002-12-18
50090-6142 KETOCONAZOLE ketoconazole A-S Medication Solutions TABLET 2020-04-10
50090-7538 Ketoconazole Ketoconazole A-S Medication Solutions SHAMPOO, SUSPENSION 2025-02-07
51407-279 Ketoconazole Ketoconazole Golden State Medical Supply, Inc. CREAM 2002-12-18
51672-1298 Ketoconazole Ketoconazole Sun Pharmaceutical Industries, Inc. CREAM 2002-12-18
51672-4026 Ketoconazole Ketoconazole Sun Pharmaceutical Industries, Inc. TABLET 1999-06-15
55505-192 Nizoral Ketoconazole Kramer Laboratories SHAMPOO 2019-01-07
55505-196 Nizoral Ketoconazole Kramer Laboratories SHAMPOO 2022-06-16
55505-232 Nizoral Ketoconazole Kramer Laboratories SHAMPOO 2025-10-01
55505-233 Nizoral Ketoconazole Kramer Laboratories SHAMPOO 2024-11-01
60429-020 Ketoconazole Ketoconazole Golden State Medical Supply, Inc. TABLET 1999-06-15
63187-774 Ketoconazole Ketoconazole Proficient Rx LP CREAM 2002-12-18
63629-8675 Ketoconazole Ketoconazole Bryant Ranch Prepack SHAMPOO, SUSPENSION 2010-01-19
63629-8676 ketoconazole ketoconazole Bryant Ranch Prepack AEROSOL, FOAM 2011-08-30
63629-8677 ketoconazole ketoconazole Bryant Ranch Prepack AEROSOL, FOAM 2011-08-30
63629-8819 Ketoconazole Ketoconazole Bryant Ranch Prepack CREAM 2019-02-08
63629-8820 Ketoconazole Ketoconazole Bryant Ranch Prepack CREAM 2019-02-08
63646-010 Ketoconazole Ketoconazole TOLMAR Inc. SHAMPOO, SUSPENSION 2005-04-11
64380-827 KETOCONAZOLE KETOCONAZOLE Strides Pharma Science Limited TABLET 2018-06-26
67296-0448 ketoconazole ketoconazole Redpharm Drug CREAM 2004-04-28
67296-0540 Ketoconazole Ketoconazole Redpharm Drug CREAM 2002-12-18
67296-1807 Ketoconazole Ketoconazole RedPharm Drug CREAM 2019-02-08
67296-2089 Ketoconazole Ketoconazole Cream, 2% RedPharm Drug CREAM 2021-05-27
68071-1709 Ketoconazole Ketoconazole NuCare Pharmaceuticals,Inc. CREAM 2002-12-18
68071-3512 Ketoconazole Ketoconazole Cream, 2% NuCare Pharmaceuticals,Inc. CREAM 2021-05-27
68788-8233 Ketoconazole Ketoconazole Cream, 2% Preferred Pharmaceuticals Inc. CREAM 2022-08-08
68788-8257 Ketoconazole Ketoconazole Preferred Pharmaceuticals Inc. SHAMPOO, SUSPENSION 2022-09-16
68788-8868 Ketoconazole Ketoconazole Preferred Pharmaceuticals Inc. SHAMPOO, SUSPENSION 2025-04-24
69292-224 Ketoconazole Ketoconazole Amici Pharma Inc. TABLET 2025-06-21
70518-4236 Ketoconazole Ketoconazole Cream, 2% REMEDYREPACK INC. CREAM 2024-12-05
70685-001 Ketoconazole Ketoconazole Esjay Pharma LLC TABLET 2025-09-10
70700-160 Ketoconazole Ketoconazole Foam Xiromed, LLC AEROSOL, FOAM 2021-05-21
70771-1874 Ketoconazole Ketoconazole Zydus Lifesciences Limited SHAMPOO 2025-03-08
70954-662 Ketoconazole Ketoconazole ANI Pharmaceuticals, Inc. SUSPENSION 2024-09-16
71205-105 Ketoconazole Ketoconazole Proficient Rx LP SHAMPOO, SUSPENSION 2016-10-01
71335-0439 Ketoconazole Ketoconazole Bryant Ranch Prepack TABLET 1999-06-15
71335-1849 KETOCONAZOLE ketoconazole Bryant Ranch Prepack TABLET 2020-04-10
71713-097 Ketoconazole Ketoconazole THIRTY MADISON INC SHAMPOO, SUSPENSION 2005-04-11
72162-1409 Ketoconazole Ketoconazole Bryant Ranch Prepack SHAMPOO, SUSPENSION 2010-01-19
72162-1417 ketoconazole ketoconazole Bryant Ranch Prepack AEROSOL, FOAM 2011-08-30
72189-180 KETOCONAZOLE KETOCONAZOLE Direct Rx TABLET 2021-02-24
72189-422 Ketoconazole Cream Ketoconazole Cream Direct_Rx CREAM 2023-02-07
72189-428 Ketoconazole Ketoconazole Direct_Rx TABLET 2023-03-01
72578-156 Ketoconazole Ketoconazole Viona Pharmaceuticals Inc SHAMPOO 2025-03-08
72789-052 KETOCONAZOLE KETOCONAZOLE PD-Rx Pharmaceuticals, Inc. TABLET 2018-06-26
73076-182 iShanCare Balanitis Cleansing iShanCare Balanitis Cleansing Shenzhen Ishan Technology Co., Ltd SOAP 2025-02-01
82804-091 Ketoconazole Ketoconazole Cream, 2% Proficient Rx LP CREAM 2021-05-27
83364-005 FungiFree Nail Fungus Treatment Ketoconazole, Tolnaftate YITONGBADA (SHENZHEN) INTERNATIONAL TRADE CO., LTD SOLUTION 2024-05-16
83887-004 Pureskin Scalp Protection anti dandruff shampoo. Pureskin Scalp Protection anti dandruff shampoo Changsha Beiliang E-commerce Co., Ltd SHAMPOO 2025-02-03
83887-005 DERPHEA Advanced Scalp Shampoo. Advanced Scalp Shampoo Changsha Beiliang E-commerce Co., Ltd SHAMPOO 2025-02-20
84277-5665 Danil Danil compound ketoconazole solution for scalp disorders. Jiangsu Chenpai Bond Pharmaceutical Co.,Ltd. SOLUTION 2024-05-01
84277-5666 Danil Danil compound ketoconazole solution for scalp disorders. Jiangsu Chenpai Bond Pharmaceutical Co.,Ltd. LOTION 2024-05-01
84558-005 1% ketoconazole anti dandruff 1% ketoconazole anti dandruff shampoo GUANGZHOU YUSONG FINE CHEMICLS Co., Ltd SHAMPOO 2024-12-04
84659-9040 Vixa Skineal Vixa Skineal Compound ketoconazole Yunnan Yuyao Bio-pharmaceutical Co.,Ltd. CREAM 2024-06-01
84745-002 POAGCI Ketoconazole VCP-KAD001 Ketoconazole Vince (Guangzhou) Cosmetics Co., Ltd. LIQUID 2024-10-11
85384-0001 1% ketoconazole Ketoconazole TAGRID LLC SHAMPOO 2025-03-31
85384-0002 Tagrit Antifungal Treament Ketoconazole 1% Ketoconazole TAGRID LLC CREAM 2025-04-18
85521-001 dandRX 1% Ketoconazole Anti-Dandruff dandRX 1% Ketoconazole Anti-Dandruff Shampoo dandRX LLC LIQUID 2025-04-09

 Mechanism of Action Classification 

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